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11 天
WWZ-11-098的发现:一种高效且具有选择性的CDK6降解剂
靶向CDK6降解剂WWZ-11-098的设计与抗肿瘤活性研究。该化合物通过优化PROTAC结构,实现高效CDK6降解(DC50=2.6nM,Dmax>99%),选择性 ...
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